Neurotransmitter receptor binding and drug discovery

J Med Chem. 1983 Dec;26(12):1667-72. doi: 10.1021/jm00366a001.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • 2-Chloroadenosine
  • Adenosine / analogs & derivatives
  • Adenosine / metabolism
  • Animals
  • Barbiturates / metabolism
  • Binding, Competitive
  • Diazepam / metabolism
  • Phenylisopropyladenosine / metabolism
  • Receptors, Drug / metabolism*
  • Receptors, GABA-A
  • Receptors, Neurotransmitter / metabolism*
  • Receptors, Purinergic
  • Xanthines / metabolism
  • gamma-Aminobutyric Acid / metabolism

Substances

  • Barbiturates
  • Receptors, Drug
  • Receptors, GABA-A
  • Receptors, Neurotransmitter
  • Receptors, Purinergic
  • Xanthines
  • 2-Chloroadenosine
  • Phenylisopropyladenosine
  • 1,3-diethyl-8-phenylxanthine
  • gamma-Aminobutyric Acid
  • Adenosine
  • Diazepam